1. “2-Oxoesters compounds and uses thereof” G. Kokotos, E. A. Dennis, WO2016/128132.
2. “Beta-lactones inhibitors of phospholipase A2 and uses thereof” G. Kokotos, E. A. Dennis, WO2016/128131.
3. “Autotaxin inhibitors and uses thereof” G. Kokotos, PCT/EP2016/000805.
4. “2-Oxothiazole compounds having activity as cPLA2 inhibitors for the treatment of anti-inflammatory disorders and hyperproliferative disorders” B. Johansen, M. Sanderberg, I.-R. Aukrust, G. Kokotos, J. Evenas, T. Brimert, G. Kildhal-Andersen, WO2016/016472A1.
5. “Antiinflammatory and antitumor 2-oxothiazoles and 2-oxothiophenes” B. Johansen, M. Sanderberg, I.-R. Aukrust, G. Kokotos, E. Barbayianni, WO2014118195-A1.
6. “2-Oxoamide inhibitors of phospholipase A2 activity and cellular arachidonate release based on dipeptides and pseudopeptides” E. A. Dennis, G. Kokotos, V. Constantinou-Kokotou, US 8,580,852, 2013.
7. “PYRROLIDINE-THIOXOPYRIMIDINONE/THIOHYDANTOIN ORGANOCATALYSTS” G. Kokotos, C. G. Kokotos, D. Limnios, EP10386007.8 (19/3/2010).
8. “ANTI INFLAMMATORY 2-OXOTHIAZOLES AND 2-OXOOXAZOLES” G. Kokotos, B. Johansen, V. Magrioti, M. Tsakos, PCT/EP2010064687.
9. “AMIDES AS INHIBITORS OF HUMAN SECRETED PHOSPHOLIPASE A2” E. A. Dennis, G. Kokotos, V. Constantinou-Kokotou, S. David, WO/2010/011686.
10. “PHOSPHOLIPASE A2 INHIBITORS AND THEIR USE IN TREATING NEUROLOGICAL INJURY AND DISEASE” E.A. Dennis, D. Stephens, S. David, R. Lopez-Vales, A. Kalyvas, G. Kokotos, V. Constantinou-Kokotou. E. Barbayianni, V. Magrioti, WO 2009009449 A2, 2009-01-15.
11. “PERFLUOROKETONE COMPOUNDS AND USES THEREOF” S. David, A. Kalyvas, R. Lopez, G. Kokotos, V. Constantinou-Kokotou, C. Baskakis, C. G. Kokotos, D. Stephens, E. A. Dennis, WO 2008122119 A1, 2008-10-16.
12. “SYSTEMIC AND INTRATHECAL EFFECTS OF A NOVEL SERIES OF PHOSPHOLIPASE A2 INHIBITORS ON HYPERALGESIA AND SPINAL PGE2 RELEASE” E.A. Dennis, T. Yaksh, K. K. Lucas, C. Svensson, D.A. Six, G. Kokotos, V. Constantinou-Kokotou, WO 2007/022443 A2.
13. “MONOESTERS AND MONOETHERS OF 2-AMINO-GLYCEROL CONTAINING LONG CHAINS AND STRUCTURALLY RELATED COMPOUNDS: PREPARATION AND USE” G. Kokotos, V. Constantinou-Kokotou, GR 20050100169 A, 2006-11-23.
14. “NOVEL ANTIHYPERTENSIVE PRODUCTS” T. Mauromoustakos, G. Kokotos, P. Mourtaveli-Minakakis, GR 1004905 B1, 2005-05-27.
15. “COMPOSITIONS AND METHODS FOR INHIBITION OF PHOSPHOLIPASE A2 MEDIATED INFLAMMATION” E. A. Dennis, T. Yaksh, K. K. Lucas, C. Svensson, D. A. Six, G. Kokotos, V. Constantinou-Kokotou, WO 03076389 A1, 2003-09-18.
16. “2-AMINO-ALKANOIC ACID DERIVATIVES, 2-AMINO ALCOHOLS AND DIAMINES, THE PROCESSES FOR THEIR PREPARATION AND THEIR USES” V. Martin, G. Kokotos, GB 2323594 A, 1998-09-30.